I-Tiamulin Hydrogen Fumarate(55297-96-6)
Incazelo Yomkhiqizo
● I-Tiamulin hydrogen fumarate isetshenziselwa isifo sokuphefumula esingapheli ezinkukhuni, i-Mycoplasma pneumonia ne-Haemophilus pleuropneumonia ezingulubeni, kanye nesifo sohudo esibangelwa i-Leptospira densa ezingulubeni.
● Izici: i-crystalline powder emhlophe noma ephuzi;enephunga elincane lesici.Incibilika emanzini (6%), umkhiqizo owomile uzinzile futhi ungagcinwa iminyaka emi-5 ngaphansi kophawu.
● I-Tiamulin hydrogen fumarate isetshenziselwa isifo sokuphefumula esingapheli ezinkukhuni, i-Mycoplasma pneumonia ne-Haemophilus pleuropneumonia ezingulubeni, kanye nesifo sohudo esibangelwa i-Leptospira densa ezingulubeni.
● I-Tiamulin fumarate inomsebenzi omuhle wokulwa namagciwane ngokumelene nezinhlobonhlobo ze-cocci e-gram-positive kuhlanganise neningi le-staphylococci ne-streptococci (ngaphandle kwe-group D streptococci) kanye nezinhlobonhlobo ze-mycoplasma namanye ama-spirochetes.Kodwa-ke, inomsebenzi we-antibacterial obuthakathaka ngokumelene namagciwane athile angalungile, ngaphandle kwe-Haemophilus spp.kanye nezinhlobo ezithile ze-Escherichia coli ne-Klebsiella.
Into | Ukucaciswa | Umphumela |
Ukubukeka | I-crystal powder emhlophe noma cishe emhlophe | Iyahambisana |
Ukuhlonza | I-HPLC: Isikhathi sokugcina esitholwe kusixazululo sokuhlola esihambisana nalokho okutholwe kusixazululo esijwayelekile | 0.2% 0.06% |
IR: I-IR yesampula ehambisana nalelo zinga eliyisethenjwa | Iyahambisana | |
Umbala nokucaca kwesixazululo | Isixazululo kufanele sicace futhi singabi nambala, futhi ukumuncwa ku-400nm naku-650nm akukukhulu kuno-0.150 no-0.030 | 99.8% |
Ukuzungezisa okuqondile | + 24 ~ 28° | Iyahambisana |
PH | 3.1~4.1 | 0.12%~0.09% |
Ukulahlekelwa ekomisweni | ≤ 0.5% | Iyahambisana |
Iphoyinti lokuncibilika | 143–149°C | 0.05ppm |
Okuqukethwe kwe-Fumarate | 83.7 ~ 87.3mg | 0.05ppm |
Izinsalela ekushiseni | ≤ 0.1% | 0.05ppm |
Izinsimbi ezinzima | ≤ 0.001% | Iyahambisana |
Izinsalela ze-solvent | ≤ 0.5% | Iyahambisana |
Ubumsulwa beChromatographic | Noma yikuphi ukungcola okuhlonziwe ≤ 1.0% | |
Noma yikuphi ukungcola okungaziwa ≤ 0.5% | Iyahambisana | |
Ukungcola okuphelele≤ 2.0% | Iyahambisana | |
I-Assay (eyomisiwe) | 98.0~102.0% | Iyahambisana |
I-Salmonella | Okubi | Iyahambisana |